氢氯噻嗪的药物-药物共结晶研究

81402898
2014
H3410.药物分析
王建荣
青年科学基金项目
高级工程师
中国科学院上海药物研究所
23万元
药物-药物共结晶;氢氯噻嗪;高通量筛选;联合用药;固态化学
2015-01-01到2017-12-31
  • 中英文摘要
  • 结题摘要
  • 结题报告
  • 项目成果
  • 项目参与人
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序号 标题 类型 作者
1 甜菊双糖苷晶型A、其制备方法、食品组合物及应用 专利 朱理平;梅雪锋;黄颖;王建荣
2 醋酸曲安奈德晶型B、其制备方法、包含所述晶型B的药物组合物和用途 专利 梅雪锋;王建荣;朱冰清;鲍俊杰
3 Structure, physicochemical properties and pharmacokinetics of resveratrol and piperine cocrystals 期刊论文 He Hongyan;Zhang Qi;Wang Jian-Rong;Mei Xuefeng
4 Mechanochromism triggered fluorescent color switching among polymorphs of a natural fluorescence pigment 期刊论文 Li Meiqi;Zhang Qi;Wang Jian-Rong;Mei Xuefeng
5 Pharmaceutical cocrystals of the anti-tuberculosis drug pyrazinamide with dicarboxylic and tricarboxylic acids 期刊论文 Wang Jian-Rong;Ye Chanjuan;Zhu Bingqing;Zhou Chun;Mei Xuefeng
6 Vapor triggered fluorescent color changes among solvates of Emodin 期刊论文 Li Meiqi;Zhang Qi;He Hongyan;Wang Jian-Rong;Mei Xuefeng
7 A new polymorph of 1-hydroxy-2-naphthoic acid obtained during failed co-crystallization experiments 期刊论文 Zhang Qi;Li Meiqi;Mei Xuefeng
8 吡咯并喹啉醌的二钠盐结晶 专利 朱理平;陆鹂烨;王建荣;孙琳琳;梅雪锋;顾建新
9 Selective crystallization of vitamin D3 for the preparation of novel conformational polymorphs with distinctive chemical stability 期刊论文 Wang Jian-Rong;Zhu Bingqing;Yu Qihui;Mei Xuefeng
10 Improving the dissolution and bioavailability of 6-mercaptopurine via co-crystallization with isonicotinamide. 期刊论文 Wang Jian-Rong;Yu Xueping;Zhou Chun;Lin Yunfei;Chen Chen;Pan Guoyu;Mei Xuefeng
11 制备高结晶度、粒径大的肌醇的结晶工艺及应用 专利 朱理平;梅雪锋;黄颖;王建荣
12 一种淫羊藿苷H1晶型、其制法和其药物组合物与应用 专利 朱理平;梅雪锋;贾丽娜;王建荣;张奇
13 一种黄芩素γ晶型、其制法和其药物组合物与用途 专利 朱理平;梅雪锋;朱冰清;王建荣
14 一种黄芩苷A晶型、其制备方法及其应用 专利 朱理平;梅雪锋;王建荣;王晓娟;朱冰清
15 Polymorphism observed in dapsone-flavone cocrystals that present pronounced differences in solubility and stability 期刊论文 He Hongyan;Jiang Linglei;Zhang Qi;Huang Ying;Wang Jian-Rong;Mei Xuefeng
16 Isostructurality in six celecoxib co-crystals introduced by solvent inclusion 期刊论文 Wang Xiaojuan;Zhang Qi;Jiang Linglei;Xu Yun;Mei Xuefeng
17 Two New Polymorphs of Huperzine A Obtained from Different Dehydration Processes of One Monohydrate 期刊论文 Zhang Qi;Mei Xuefeng
18 Drug-drug co-crystallization presents a new opportunity for the development of stable vitamins 期刊论文 Wang Jian-Rong;Yu Qihui;Dai Wenjuan;Mei Xuefeng
19 甜菊糖C苷晶型V、其制备方法、食品组合物及应用 专利 朱理平;梅雪锋;黄颖;王建荣
20 吡咯并喹啉醌的二钠盐结晶 专利 朱理平;陆鹂烨;王建荣;孙琳琳;梅雪锋;顾建新
21 一种淫羊藿苷Form α晶型、其制法和其药物组合物与应用 专利 朱理平;梅雪锋;贾丽娜;王建荣;张奇
22 固体药物的转晶现象 期刊论文 张奇;梅雪锋
23 pH-Switchable vitamin B9 gels for stoichiometry-controlled spherical co-crystallization. 期刊论文 Wang Jian-Rong;Bao Junjie;Fan Xiaowu;Dai Wenjuan;Mei Xuefeng
24 一种淫羊藿苷H2晶型、其制法和其药物组合物与应用 专利 朱理平;梅雪锋;贾丽娜;王建荣;张奇
25 Insight into the Phase Transformation among Various Solid Forms of Baicalein 期刊论文 Zhu Bingqing;Wang Jian-Rong;Mei Xuefeng
26 Absolute asymmetric synthesis of a sanguinarine derivative through crystal-solution interactions 期刊论文 Zhang Qi;Jia Lina;Wang Jian-Rong;Mei Xuefeng
27 Determination of absolute configuration using heavy atom based co-crystallization method: Halogen atom effects 期刊论文 Wang Jian-Rong;Fan Xiaowu;Ding Qiaoce;Mei Xuefeng
28 Taming photo-induced oxidation degradation of dihydropyridine drugs through cocrystallization. 期刊论文 Yu Qihui;Yan Zhicheng;Bao Junjie;Wang Jian-Rong;Mei Xuefeng
29 甜菊糖B苷晶型G、其制备方法、食品组合物及应用 专利 朱理平;梅雪锋;黄颖;王建荣
30 Improving Dissolution and Photostability of Vitamin K3 via Cocrystallization with Naphthoic Acids and Sulfamerazine 期刊论文 Zhu Bingqing;Wang Jian-Rong;Zhang Qi;Mei Xuefeng
31 缬沙坦晶型E的诱导结晶工艺及应用 专利 朱理伟;梅雪锋;黄颖;王建荣
32 甜菊糖B苷钠盐晶型A、其制备方法、食品组合物及应用 专利 朱理平;梅雪锋;黄颖;王建荣
33 吡咯并喹啉醌的二钠盐结晶 专利 朱理平;陆鹂烨;王建荣;孙琳琳;梅雪锋;顾建新
34 一种甜菊糖D苷晶型A、其制备方法及其应用 专利 朱理平;梅雪锋;黄颖;王建荣;张奇
35 Amino acids as co-amorphous excipients for tackling the poor aqueous solubility of valsartan 期刊论文 Huang Ying;Zhang Qi;Wang Jian-Rong;Lin Kai-Lei;Mei Xuefeng
36 Zwitterionic Cocrystals of Flavonoids and Proline: Solid-State Characterization, Pharmaceutical Properties, and Pharmacokinetic Performance 期刊论文 He Hongyan;Huang Ying;Zhang Qi;Wang Jian-Rong;Mei Xuefeng
37 Solid-state characterization of 17 beta-estradiol co-crystals presenting improved dissolution and bioavailability 期刊论文 Wang Jian-Rong;Wang Xiaojuan;Yang Yong;Chen Xiaoyan;Mei Xuefeng
38 Modulating the Dissolution and Mechanical Properties of Resveratrol by Cocrystallization 期刊论文 He Hongyan;Zhang Qi;Li Meiqi;Wang Jian-Rong;Mei Xuefeng
39 替米沙坦与氢氯噻嗪的共晶 专利 王建荣
40 Versatile solid modifications of icariin: structure, properties and form transformation 期刊论文 Jia Lina;Zhang Qi;Wang Jian-Rong;Mei Xuefeng
41 大黄素晶型Ι、其制备方法、药物组合物及应用 专利 朱理平;梅雪锋;李美琪;王建荣;张奇
42 Polymorphs and Hydrates of Apatinib Mesylate: Insight into the Crystal Structures, Properties, and Phase Transformations 期刊论文 Zhu Bin;Wang Jian-Rong;Ren Guobin;Mei Xuefeng
43 甜菊糖M苷晶型及制备方法和用途 专利 朱理平;梅雪锋;黄颖;王建荣
44 Polymorphism of Triamcinolone Acetonide Acetate and Its Implication for the Morphology Stability of the Finished Drug Product 期刊论文 Wang Jian-Rong;Zhu Bingqing;Zhang Zaiyong;Bao Junjie;Deng Gaojin;Ding Qiaoce;Mei Xuefeng
45 Cocrystals of Baicalein with Higher Solubility and Enhanced Bioavailability 期刊论文 Zhu Bingqing;Zhang Qj;Wang Jian-Rong;Mei Xuefeng
46 Insight into the conformational polymorph transformation of a block-buster multiple sclerosis drug fingolimod hydrochloride (FTY 720) 期刊论文 Wang Jian-Rong;Li Sha;Zhu Bingqing;Mei Xuefeng
47 Greener solid-state synthesis: stereo-selective [2+2] photodimerization of vitamin K-3 controlled by halogen bonding 期刊论文 Zhu Bingqing;Wang Jian-Rong;Zhang Qi;Mei Xuefeng
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