【20872071】Ugi反应合成新型绿色杀菌剂甲噻酰胺的衍生物及其生物活性研究国家自然基金项目

Ugi反应合成新型绿色杀菌剂甲噻酰胺的衍生物及其生物活性研究

项目批准号： 20872071

批准年份： 2008

学科分类： B0706.药物化学生物学

项目负责人：范志金

资助类别：面上项目

负责人职称：教授

依托单位：南开大学

资助金额： 33万元

关键词： Ugi反应;3-噻二唑;1;平行合成;2;甲噻酰胺

起止时间： 2009-01-01到2011-12-31

中英文摘要
结题摘要
结题报告
项目成果
项目参与人

查看更多信息请先登录或注册

序号	标题	类型	作者
1	Synthesis, crystal structure and biological activity of N-tert-butyl-N-(4-methyl-1,2,3-thiadiazole)-5-yl-N'-(4-methyl-1,2,3-thiadiazole)-5-formyl-N'-3,5-dichloropyridin-2-yl-diacylhydrazine	期刊论文	Zhang You-Jun\|Song Hai-Bin\|Fu Yi-Feng\| Belskaya N. P.\|Bakulev V. A.\|Wu Qing-Jun\|Wang Huan\|Fan Zhi-Jin\|
2	Synthesis and insecticidal activity of N-tert-butyl-N,N′- diacylhydrazines containing 1,2,3-thiadiazoles	期刊论文	Wang Huan\|Zhang Zhengcai\|Liu Feng\|Yang Zhikun\|Song Haibin\|Mi Na\|Wu Qingjun\|Wang Shouxin,\|Fan Zhijin\|Zhang Youjun\|
3	植物激活剂作用机制的初步研究	会议论文	王盾\|范志金\|李岳东\|黄杰\|国丹丹\|华学文\|姬晓恬\|房震\|赵晖\|范谦\|
4	基于植物诱导抗病激活机制的先导优化和生物活性研究	会议论文	Belskaya N. P.\|Prokhorova P. E.\|Vasiliy A. Bakulev.\|Morzherin Yu. Yu.\|赵晖\|王守信\|国丹丹\|王唤\|范志金\|黄杰\|房震\|李岳东\|
5	鱼尼丁受体类杀虫剂的研究进展	期刊论文	王唤\|米娜\|Bakulev V. A.\|Belskaya N. P.\|范志金\|
6	Two directions for the oxidative heterocyclization of arylhydrazonoacetamidines	会议论文	N. P. Belskaya\|N. Mi\|V. A. Bakulev\|E. N. Akhtarieva\|Z. Fan\|S. G. Lesogorova\|
7	《农药学学报》创刊十周年 10 篇优秀论文	奖励	李正名\|范志金\|王玲秀\|钱传范\|陈俊鹏\|
8	新型植物激活剂创制的基础研究	会议论文	王唤\|Vasiliy A. Bakulev\|米娜\|马琳\|范志金\|范志银\|杨知昆\|郑琴香\|张海科\|左翔\|
9	Molecular Design, Synthesis and biological sctivity of novel 1,2,3-thiadiazoles	会议论文	Na Mi\|Zhijin Fan\|Huan Wang\|Shouxin Wang\|Yifeng Fu\|Dandan Guo\|Hui Zhao\|
10	Synthesis and Crystal Structure of 3,6-Bis(4-methyl-1,2,3-thiadiazol-5-yl)-1,2,4-triazolo[3,4-b] [1,3,4]thiadiazole	期刊论文	Vasiliy, A. Bakulev\|Zuo Xiang\|Yang Zhi-Kun\|Zheng Qin-Xiang\|Song Hai-Bin\|Natalia, P. Belskaia\|Fan Zhi-Jin\|You Jin-Mao\|
11	杀菌剂氟菌螨酯及其中间体的HPLC分析	期刊论文	李淑芹\|蔡飞\|范志金\|王海英\|刘长令\|陈建宇\|李申\|
12	Synthesis, crystal structure, and biological activity of naphthalen-2-yl-4-methyl-1,2,3-thiadiazole-5-carboxylate	期刊论文	Mi Na\|Fu Yi-Feng\|Wang Shou-Xin\|Fan Zhi-Jin\|Bakulev Vasiliy A.\|Song Hai-Bin\| Belskaya Nataliya P.\|Zhang Hai-Ke\|
13	Synthesis of 4-methyl-1,2,3-thiadiazole derivatives via Ugi reaction and their biological activities	期刊论文	Na Mi\|Huan Wang\|Zhikun Yang\|Xiang Zuo\|Haike Zhang\|Qingxiang Zheng\|Zhijin Fan\|
14	三唑并噻二唑衍生物的合成及抑菌活性	期刊论文	米娜\|张海科\|孙学军\|杨知昆\|范志金\|尤进茂\|
15	三唑类化合物的研究进展及其在新农药创制中的应用	会议论文	房震\|范志金\|范谦\|赵晖\|国丹丹\|米娜\|李岳东\|
16	Synthesis and biological activity of novel 1,2,3-thiadiazoles	会议论文	Yifeng Fu\|Shouxin Wang\|Dandan Guo\|Huan Wang\|Haike Zhang\|Zhijin Fan\|Na Mi\|Zhikun Yang\|Hui Zhao\|
17	Synthesis and Biological Activity Evaluation of 1,2,3-Thiadiazole Derivatives as Potential Elicitors with Highly Systemic Acquired Resistance	期刊论文	Liu, Xiufeng\|Zuo, Xiang\|Ma, Lin\|Zhang, Haike\|Zheng, Qinxiang\|Mi, Na\|Shi, Zugui\|Bao, Lili\|Fan, Zhijin\|
18	鱼尼汀受体类杀虫剂的研究进展	会议论文	范志金\|王唤\|郑琴香\|张海科\|杨知昆\|左翔\|马琳\|米娜\|
19	异噻唑类化合物的研究进展	会议论文	赵晖\|姬晓恬\|李岳东\|范志金\|房震\|国丹丹\|华学文\|
20	Synthesis and Biological Activity of Organotin 4-Methyl-1,2,3-thiadiazole-5-carboxylates and Benzo[1,2,3]thiadiazole-7-carboxylates	期刊论文	Ma, Lin\|Fan, Zhi-Jin\|Wang, Zhi-Hong\|Zhang, Jun\|Guo, Yan-Zhao\|Song, Hai-Bin\|
21	4-Methyl-1,2,3-thiadiazoles synthesized via Ugi reaction with antiviral activity against tobacco mosaic virus	期刊论文	Huang Jie\|Fu Yifeng,\|Mi Na\|Huang Yun\|Wang Huan\|Zheng Qingxiang\|Bakulev V. A.\|Belskaya N. P.\|Fan Zhi-Jin \|Zuo Xiang\|
22	Discovery of methiadinil as novel candidate plant elicitor	会议论文	Lin Ma\|Huan Wang\|Na Mi\|Zhikun Yang\|Xiang Zuo\|Haike Zhang\|Zhijin Fan\|Qingxiang Zheng\|Zugui Shi\|
23	Synthesis of 3,5-dichloro-4-(1,1,2,2- tetrafluoroethoxy) phenyl containing 1,2,3-thiadiazole derivatives via Ugi reaction and their biological activities	期刊论文	Shouxin Wang\|Nataliya P. Belskaya\|Zhengcai Zhang\|Yifeng Fu\|Huan Wang\|Na Mi\|Jufang Zhang\|Vasiliy A. Bakulev.\|Zhijin Fan\|
24	2-Hydroxypropyl derivatives of 1,2,3 thiadiazole and 1,2,3-triazole: Synthesis and antifungal activity	期刊论文	Yury Morzherin\|Polina E. Prokhorova\|Dmitry A. Musikhin\|Zhijin Fan\|Tatiana V. Glukhareva\|
25	Wq-C-13的生物活性和作用机制的初步研究	会议论文	范志金\|黄杰\|张海科\|吴琼\|付一峰\|米娜\|范谦\|房震\|
26	基于多组分 Ugi 反应的植物激活剂先导优化和生物活性研究	会议论文	贾俊超\|左翔\|米娜\|王唤\|杨知昆\|马琳\|吴琼\|张海科\|范志金\|郑琴香\|
27	5-Methyl-1,2,3-thiadiazoles synthesized via Ugi reaction and their fungicidal and antiviral activity	期刊论文	Yang, Z. K. \| Zhang, H. K.\|Mi, N.\|Fan Z. J.\|Wang, H.\|Zuo, X.\|Zheng, Q. X.\|
28	Synthesis and reactions of thioamides of 5-amino-2-aryl-2H-1,2,3-triazole-4- carboxylic acid	期刊论文	Eltsov, O. S.\|Sapozhnikova, S. G.\|Belskaya, N. P.\|Bakulev, V. A.\|Slepukhin, P. A.\|Fan, Z. -J.\|
29	基于1,2,3-噻二唑的双酰肼衍生物的设计合成和生物活性	会议论文	范志金\|王唤\|李岳东\|黄杰\|王守信\|赵晖\|房震\|国丹丹\|
30	Basic Studies on the Development of Novel Plant Elicitor	会议论文	Zhijin Fan\|Lili Bao\|Zugui Shi,\|Xiang Zuo\|Fengli Liu\|Haike Zhang\|Qiong Wu\|Zhikun Yang\|Lin Ma\|Xiufeng Liu\|
31	环糊精及其衍生物在农药领域应用的研究进展	期刊论文	张晓光\|王海英\|范志金\|刘洁翔\|
32	Methiadinil, a novel candidate plant elicitor for crop protection	会议论文	Zhijin Fan\|Zugui Shi\|Qian Fan\|Zhikun Yang\|Na Mi\|Huan Wang\|Lin Ma\|Xiang Zuo\|Haike Zhang\|Xuelin Chen\|Qingxiang Zheng\|
33	Synthesis, structure and biological activity of triorganotin 1H-tetrazolyl-1-acetates: cyclic hexamer and linkage coordination polymers	期刊论文	Xie, Yun-Fu\|Ma, Lin\|Fan, Zhi-Jin\|Mi, Na\|Tang, Liang-Fu\|Yu, Yang\|
34	4-甲基-1,2,3-噻二唑-5-甲酸芳酯的合成及生物活性	期刊论文	范志金\|张聚方\|宋海斌\|张正财\|BELSKAYA N.P.\|BAKULEV V.A.\|米娜\|王守信\|付一峰\|王唤\|黄云\|
35	苯甲酰脲类杀虫剂研究进展	会议论文	杨知昆\|王唤\|张海科\|郑琴香\|范志金\|左翔\|马琳\|米娜\|
36	具有诱导抗病活性的农药先导设计和生物活性	会议论文	黄杰\|姬晓恬\|赵晖\|Vasiliy A. Bakulev\|李岳东\|国丹丹\|华学文\|王盾\|范志金\|房震\|Tatiana A. Kalinina\|
37	具有生物活性的N-苯基-N'-(1,3-噻唑-2-基)-1,2,3-苯并噻二唑-7-甲脒的晶体结构与理论计算	期刊论文	范志金\|徐布一\|鲍丽丽\|李权\|赵可清\|
38	Synthesis, crystal structure and biological activity of two 1,2,3-thiadiazole derivatives	期刊论文	Wang Shou-Xin\|Fan Zhi-Jin\|Bakulev Vasiliy A.\|Fu Yi-Feng\|Song Hai-Bin\|Zhang Zheng-Cai\|Wang Huan\|Huang Jie\|Belskaya Nataliya P.\|Mi Na\|
39	阿维菌素水乳剂的稳定性	期刊论文	王满意\|范志金\|张晓光\|王海英\|刘洁翔\|
40	Synthesis, Crystal Structure and Biological activity of N′-tert-butyl-N-(3-methoxylbenzoyl)- N-(4-methyl-1,2,3-thiadiazole-5-formyl hydrazine	期刊论文	Yun Huang\|Polina E. Prokhorova\|Nataliya P. Belskaya\|Zhi-Jin Fan\|Yury Yu. Morzherin\|Hai-Bin Song\|Hui Zhao\|Jie Huang\|Vasiliy A. Bakulev\|Huan Wang\|
41	1,2,3-噻二唑联-1,2,4-三唑衍生物的合成及抑菌活性	期刊论文	孙学军\|范志金\|Vasiliy A.Bakulev\|尤进茂\|张海科\|Natalia P.Belskaia\|米娜\|宋海斌\|杨知昆\|
42	苯甲酰脲类杀虫剂研究进展	期刊论文	张海科\|王唤\|Vasiliy A.Bakulev\|Natalia P.Belskaia\|范志金\|米娜\|
43	Bitriazolyl acyclonucleosides synthesized via Huisgen reaction using internal alkeynes show antiviral activity tobacco mosaic virus	期刊论文	Zhijin Fan\|Liang Feng\|Yifeng Fu\|Yi Xia\|Alain Maggiani\|Ling Peng\|Menghua Wang\|Jianhua Yao\|Ruizhi Zhu\|Fanqi Qu\|
44	Synthesis, crystal structure, and biological activity of 4-methyl-1,2,3- thiadiazole containing 1,2,4-triazolo-[3,4-b][1,3,4]-thiadiazoles.	期刊论文	Song, Haibin\|Yang, Zhikun\|Zhijin, Fan\|Xiang, Zuo\|Wang, Huan\|Zheng, Qinxiang\|Mi, Na\|Zhang, Haike\|Cai, Fei\|
45	新型杀菌剂异噻菌胺	会议论文	王盾\|黄云\|陈晓燕\|范志金\|黄杰\|
46	Lead derivation and biological activity of plant elicitor.	会议论文	Natalia P. Belskaia\|Qinxiang Zheng\|Hui Zhao\|Vasiliy A. Bakulev\|Xiang Zuo\|Zhijin Fan\|Na Mi\|Huan Wang\|
47	BASF Excellent Poster Award at The 1st China-Japan-Korea Workshop on Pesticide Science in Shanghai China	奖励	Xiufeng Liu\|Lili Bao\|Fengli Liu\|Zugui Shi\|Lin Ma\|Xiang Zuo\|Qiong Wu\|Zhikun Yang\|Fan Zhijin\|Haike Zhang\|

查看更多信息请先登录或注册

再问科研

相关项目

趋势报告

经验分享