病原细菌多胺信号转导系统抑制剂的设计与合成

31570122
2015
C0108.病原细菌学
崔紫宁
面上项目
教授
华南农业大学
62万元
合成;多胺信号转导系统;分子设计;III型分泌系统;抑制剂
2016-01-01到2019-12-31
  • 中英文摘要
  • 结题摘要
  • 结题报告
  • 项目成果
  • 项目参与人
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序号 标题 类型 作者
1 Novel S-thiazol-2-yl-furan-2-carbothioate derivatives as potential T3SS inhibitors against Xanthomonas oryzae on rice 期刊论文 Shan Jiang;Min He;Xu-Wen Xiang;Muhammad Adnan;Zi-Ning Cui
2 一种含噁唑环2,4-二取代吡唑类化合物及其制备方法和应用 专利 崔紫宁;李亚胜;胡德坤;田浩;刘星宇;宋高鹏
3 Synthesis and biological evaluation of acylated oligorhamnosidederivatives structurally related to mezzettiaside-6 with cytotoxic activity 期刊论文 Song Gaopeng;Li Sumei;Lei Zhiwei;Li Yibin;Li Junhua;Liao Yixian;Cui Zi-Ning
4 环二鸟苷酸信号分子抑制剂的研究进展 期刊论文 向绪稳;刘星宇;陶辉;崔紫宁;张炼辉
5 调节生物被膜化合物的研究进展 期刊论文 刘星宇;向绪稳;陶辉;崔紫宁;张炼辉
6 Design, synthesis and fungicidal activity of novel 2-substituted aminocycloalkylsulfonamides 期刊论文 Liu Caixiu;Yan Xiaojing;Wang Minlong;Qin Peiwen;Qi Zhiqiu;Ji Mingshan;Liu Xingyu;Babu P. Vijaya;Li Xinghai;Cui Zi-Ning
7 Discovery of Novel Inhibitors of Phosphodiesterase 4 with 1-phenyl-3,4-dihydroisoquinoline Scaffold: Structure-based drug design and Fragment Identification 期刊论文 Yixian Liao;Xiuhua Jia;Yongmei Tang;Sumei Li;Yipeng Zang;Lei Wang;Yongfeng Gao;Lijian Huo;Zi-Ning Cui;Gaopeng Song
8 Synthesis and Bioactivities of Novel Pyrazole Derivatives Containing 5-Phenyl-2-Furan 期刊论文 Wasim Ahmed;Xiaojing Yan;Dekun Hu;Muhammad Adnan;Riyuan Tang;Zi-Ning Cui
9 Synthesis, FungicidalActivity, and Structure Activity Relationship of β-Acylaminocycloalkylsulfonamidesagainst Botrytis cinerea 期刊论文 Liu Chun-Hui;Chen Xiao-Yuan;Qin Pei-Wen;Qi Zhi-Qiu;Ji Ming-Shan;Liu Xing-Yu;Babu P. Vijaya;Li Xing-Hai;Cui Zi-Ning
10 Synthesis and Bioactivity of Thiazolidin-2-cyanamide Derivatives against Type III Secretion System of Xanthomonas oryzae on Rice 期刊论文 Xuwen Xiang;Hui Tao;Shan Jiang;Lian-Hui Zhang;Zi-Ning Cui
11 Design and characterization of a polyamine derivative inhibiting the expression of type III secretion system in Pseudomonas aeruginosa 期刊论文 Wang Chao;Liu Xiaoling;Wang Jing;Zhou Jianuan;Cui Zi-Ning;Zhang Lian-Hui
12 一种含四氢异喹啉并氨基甲酸酯类化合物及其制备方法和应用 专利 宋高鹏;崔紫宁;李俊骅;韦著文;刘星宇
13 Synthesisand fungicidal activity of novel 2,5-disubstituted-1,3,4- thiadiazole derivativescontaining 5-phenyl-2-furan 期刊论文 Cui Zi-Ning;Li Ya-Sheng;Hu De-Kun;Tian Hao;Jiang Jia-Zhen;Wang Yuan;Yan Xiao-Jing
14 Synthesis and biological evaluation of 1,3,4-thiadiazole derivatives as type III secretion system inhibitors against Xanthomonas oryzae 期刊论文 Hui Tao;Hao Tian;Shan Jiang;Xuwen Xiang;Yinuo Lin;Wasim Ahmed;Riyuan Tang;Zi-Ning Cui
15 N’-5-(取代苯基)-2-呋喃甲酰基-5-丙基-1H-吡唑-3-甲酸乙酯类化合物及其制备方法与应用 专利 崔紫宁;胡德坤;田浩;李亚胜;宋高鹏;刘星宇
16 Small molecule inhibitors specifically targeting type III secretion system of Xanthomonas oryzae on rice 期刊论文 Hui Tao;Su-Su Fan;Shan Jiang;Xuwen Xiang;Xiaojing Yan;Lian-Hui Zhang;Zi-Ning Cui
17 Discovery of ethyl 2-nitro-3-arylacrylates molecules as T3SS inhibitor reducing the virulence of plant pathogenic bacteria Xanthomonas 期刊论文 Shan Jiang;Hui Li;Wasim Ahmed;Xuwen Xiang;Gaopeng Song;Zi-Ning Cui
18 Synthesis and Bioactivity of 1,3-Thiazolidine-2-thione Derivatives against Type III Secretion System of Xanthomonas oryzae. Bioorg 期刊论文 Hui Tao;Hao Tian;Shan Jiang;Xuwen Xiang;Wasim Ahmed;Riyuan Tang;Zi-Ning Cui
19 Synthesis and Biological Evaluation of 2,4-Disubstituted Oxazole Derivatives as Potential PDE4 Inhibitors 期刊论文 Li Ya-Sheng;Hu De-Kun;Zhao Dong-Sheng;Liu Xing-Yu;Jin Hong-Wei;Song Gao-Peng;Cui Zi-Ning
20 S-(5-取代-1,3,4-噻二唑)-(5-取代苯基)-2-呋喃硫代甲酸酯类化合物及其制备方法与应用ZL 201610382784.8 专利 崔紫宁;田浩;胡德坤;李亚胜;宋高鹏;刘星宇
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