黄酮碳苷类化合物的酶催化机制研究及新颖COX-2抑制剂的发现

82003614
2020
H3402.天然药物化学
易阳
青年科学基金项目
助理研究员
北京大学
24万元
碳糖基转移酶;黄酮碳苷化合物;量子力学;分子模拟;密度泛函理论
2021-01-01到2023-12-31
  • 中英文摘要
  • 结题摘要
  • 结题报告
  • 项目成果
  • 项目参与人
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序号 标题 类型 作者
1 Chrysin 7-O-β-D-glucuronide, a dual inhibitor of SARS-CoV-2 3CLpro and PLpro, for the prevention and treatment of COVID-19. 期刊论文 Yi Yang;Yu Rong;Xue Heng;Zhengtong Jin;Meng Zhang;Bao Yang-Oujie;Wang Zi-Long;Wei Hong-Ping;Qiao Xue;Yang Hang
2 Licorice-saponin A3 is a broad-spectrum inhibitor for COVID-19 by targeting viral spike and anti-inflammation 期刊论文 Yi Yang;Li Wenzhe;Liu Kefang;Xue Heng;Yu Rong;Zhang Meng;Bao Yang-Oujie;Lai Xinyuan;Fan Jingjing;Huang Yuxi;Wang Jing;Shi Xiaomeng;Li Junhua;Wei Hongping;Xiang Kuanhui;Li Linjie;Zhang Rong;Zhao Xin;Qiao Xue;Yang Hang;Ye Min
3 Schaftoside inhibits 3CLpro and PLpro of SARS-CoV-2 virus and regulates immune response and inflammation of host cells for the treatment of COVID-19 期刊论文 Yi Yang;Zhang Meng;Xue Heng;Yu Rong;Bao Yang-Oujie;Kuang Yi;Chai Yue;Ma Wen;Wang Jing;Shi Xiao-Meng;Li Wen-Zhe;Hong Wei;Li Jun-Hua;Muturi Elishiba;Wei Hong-Ping;Wlodarz Joachim;Roszak Szczepan;Qiao Xue;Yang Hang;Ye Min
4 Functional Characterization and Protein Engineering of a Triterpene 3-/6-/2'-O-Glycosyltransferase Reveal a Conserved Residue Critical for the Regiospecificity 期刊论文 Zhang Meng;Yi Yang;Gao Bai-Han;Su Hui-Fei;Bao Yang-Oujie;Shi Xiao-Meng;Wang Hai-Dong;Li Fu-Dong;Ye Min;Qiao Xue
5 Natural triterpenoids from licorice potently inhibit SARS-CoV-2 infection 期刊论文 Yi Yang;Li Jun-Hua;Lai Xin-Yuan;Zhang Meng;Kuang Yi;Bao Yang-Oujie;Yu Rong;Hong Wei;Muturi Elishiba;Xue Heng;Wei Hong-Ping;Li Tong;Zhuang Hui;Qiao Xue;Xiang Kuan-Hui;Yang Hang;Ye Min
6 A highly selective C-rhamnosyltransferase from Viola tricolor and insights into its mechanisms 期刊论文 Han Bo-Yun;Wang Zi-Long;Li Jun-Hao;Jin Qing;Wang Hao-Tian;Chen Kuan;Yi Yang;Agren Hans;Qiao Xue;Ye Min
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