基于MDM2/HDAC双靶抑制策略的抗肿瘤先导化合物发现和优化
序号 | 标题 | 类型 | 作者 |
---|---|---|---|
1 | Discovery of pyrazolone spirocyclohexadienone derivatives with potent antitumor activity | 期刊论文 | Wang Lei;Yang Zixuan;Ni Tianyu;Shi Wencai;Guo Yunbo;Li Keliang;Shi Anzhe;Wu Shanchao;Sheng Chunquan |
2 | 上海市科技进步二等奖 | 奖励 | 盛春泉;李剑;缪震元;董国强;张万年;吕加国;刘娜;武善超;姚建忠;毛斐 |
3 | 基于组蛋白去乙酰化酶的双靶点抑制剂研究进展 | 期刊论文 | 石安喆;武善超;盛春泉 |
4 | 一种MDM2蛋白降解靶向嵌合体及其制备方法和应用 | 专利 | 盛春泉;董国强;马俊辉;何世鹏;方宇昕;武善超;陈树强 |
5 | Natural Product Evodiamine with Borate Trigger Unit: Discovery of Potent Antitumor Agents against Colon Cancer | 期刊论文 | Li Xinglin;Wu Shanchao;Dong Guoqiang;Chen Shuqiang;Ma Zonglin;Liu Dan;Sheng Chunquan |
6 | Scaffold Hopping of Natural Product Evodiamine: Discovery of a Novel Antitumor Scaffold with Excellent Potency against Colon Cancer. | 期刊论文 | Wang Lei;Fang Kun;Cheng Junfei;Li Yu;Huang Yahui;Chen Shuqiang;Dong Guoqiang;Wu Shanchao;Sheng Chunquan |
7 | 多靶点抗肿瘤活性的吴茱萸碱衍生物及其制备方法与应用 | 专利 | 董国强;盛春泉;陈树强;鲁俊杰;黄亚辉;武善超;李育 |
8 | Homo-PROTAC mediated suicide of MDM2 to treat non-small cell lung cancer | 期刊论文 | He Shipeng;Ma Junhui;Fang Yuxin;Liu Ying;Wu Shanchao;Dong Guoqiang;Wang Wei;Sheng Chunquan |
9 | 药物合成——路线设计策略和案例解析 | 专著 | 张万年;盛春泉;缪震元;王胜正;武善超 |