IDO1/TDO双靶点小分子抑制剂的设计、合成及成药性研究
序号 | 标题 | 类型 | 作者 |
---|---|---|---|
1 | Structural Optimization and Structure−Activity Relationship Studies of 6,6-Dimethyl-4-(phenylamino)‑6H‑pyrimido[5,4‑b][1,4]oxazin- 7(8H)‑one Derivatives as A New Class of Potent Inhibitors of Pan-Trk and Their Drug-Resistant Mutants | 期刊论文 | Shulei Pan;Liting Zhang;Xinling Luo;Jinshan Nan;Wei Yang;Huachao Bin;Yang Li;Qiao Huang;Tianqi Wang;Zhiling Pan;Bo Mu;Falu Wang;Chenyu Tian;Yang Liu;Linli Li;Shengyong Yang |
2 | Discovery and structure-activity relationship studies of 1-aryl-1H-naphtho[2,3-d][1,2,3]triazole-4,9-dione derivatives as potent dual inhibitors of indoleamine 2,3-dioxygenase 1 (IDO1) and trytophan 2,3-dioxygenase (TDO). | 期刊论文 | Shulei Pan;Yangli Zhou;Qiusheng Wang;Yanlin Wang;Chenyu Tian;Tianqi Wang;Luyi Huang;Jinshan Nan;Linli Li;Shengyong Yang |