光学活性噻唑类绿色农药先导的优化及其作用机制的研究
序号 | 标题 | 类型 | 作者 |
---|---|---|---|
1 | Synthesis of Novel 3,4-Chloroisothiazole-Based Imidazoles as Fungicides and Evaluation of Their Mode of Action | 期刊论文 | Chen Lai;Zhao Bin;Fan Zhijin;Liu Xiumei;Wu Qifan;Li Hongpeng;Wang Haixia |
2 | 一类杂环三唑衍生物及其制备方法和用途 | 专利 | 范志金;陈来;李鸿鹏;李冀伟;胡文昊;刘秀梅;韩雪;特蒂安娜•卡林丽娜 |
3 | Discovery of Novel Isothiazole, 1,2,3-Thiadiazole, and Thiazole-Based Cinnamamides as Fungicidal Candidates | 期刊论文 | Chen Lai;Zhao Bin;Fan Zhijin;Hu Mengxu;Li Qing;Hu Wenhao;Li Jiwei;Zhang Jinlin |
4 | 一类含1,2,3-噻二唑的苯乙酮衍生物及其制备方法和用途 | 专利 | 范志金;房震;王盾;李岳东;姬晓恬;华学文;毛武涛;宗广宁;李凤云;李娟娟 |
5 | 林木主要蛀干害虫信息诱引技术体系构建及非化学防控集成示范 | 奖励 | 谷希树;白义川;张素芬;范志金;刘宝生 |
6 | Synthesis, Crystal Structure and Fungicidal Activity of Ethyl 2-(3-(4-Fluorobenzamido)phenyl)-4-((4-fluorobenzoyl)oxy)thiazole-5-carboxylate | 期刊论文 | Guo Xiao Feng;Su Han Xiang;Fan Zhi Jin;Sun Xue Wen;Sun Yao Zheng;Qin Zhong Xiang |
7 | Discovery of Pyruvate Kinase as a Novel Target of New Fungicide Candidate 3-(4-Methyl-1,2,3-thiadiazolyl)-6-trichloromethyl-[1,2,4]-triazolo-[3,4-b][1,3,4]-thiadizole | 期刊论文 | Bin Zhao;Sijia Fan;Zhijin Fan;Haixia Wang;Nailou Zhang;Xiaofeng Guo;Dongyan Yang;Qifan Wu;Bin Yu;Shuang Zhou |
8 | 一类4位取代噻唑酰胺衍生物及其制备方法和用途 | 专利 | 范志金;郭晓凤;苏瀚翔;赵斌;孙学文;张乃楼;杨冬燕;吴启凡;于斌;周爽;孙耀正 |
9 | 新型杀菌化合物靶标识别及其靶向候选药剂设计概述 | 期刊论文 | 赵斌;陈来;张乃楼;范志金 |
10 | 防治农林生物灾害的大型直升机智能飞防关键技术创新与应用 | 奖励 | 梁小文;王滨;郑国华;范志金;钟玲;吴学民;付恭华;曾平章;肖筱成;陈玉芹;周清 |
11 | 一类手性哌啶衍生物及其制备方法和用途 | 专利 | 范志金;朱玉洁;马刘勇;郭晓凤;陈来;钱晓琳;张乃楼;王海霞;张秩鸣;徐京华 |
12 | Approach to thiazole-containing tetrahydropyridine derivatives via Aza-Rauhut-Currier reaction and their potent fungicidal and insecticidal activity | 期刊论文 | Y.J. Zhu;X.F. Guo;Z.J. Fan;L. Chen;L. Y. Ma;H.X. Wang;Y. Wei;X.M. Xu;J.P. Lin;V. A. Bakulev |
13 | 25%甲噻诱胺悬浮剂登记证 | 奖励 | 范志金;范谦;邱丰;殷勇;员工们 |
14 | 一类3,4-二氯异噻唑-5-甲脒衍生物及其制备方法和用途 | 专利 | 范志金;宗广宁;马刘勇;李凤云;朱玉洁;陈来;王海霞;钱晓琳;郭晓凤;裴钰;徐京华 |
15 | 一类异噻唑肟醚甲氧基丙烯酸酯衍生物及其制备方法和用途 | 专利 | 范志金;陈来;郭晓凤;朱玉洁;钱晓琳;马刘勇;张乃楼;王海霞;张秩鸣;徐京华;宋胤奇 |
16 | 一类含4-甲基-1,2,3-噻二唑的4,5-二氢噻唑醇酸酯衍生物及其制备方法和用途 | 专利 | 范志金;毛武涛;刘超伦;李娟娟;姬晓恬;华学文;宗广宁;李凤云;房震;李岳东 |
17 | 一类三取代噻唑酰胺衍生物及其制备方法和用途 | 专利 | 范志金;郭晓凤;邓有才;吴启凡;张乃楼;杨冬燕;赵斌;于斌;周爽;孟勐;黄纯;王芳杰;马容基 |
18 | Synthesis and fungicidal activity of 3,4-dichloroisothiazolebased strobilurins as potent fungicide candidates | 期刊论文 | Lai Chen;Xiao-Feng Guo;Zhi-Jin Fan;Nai-Lou Zhang;Yu-Jie Zhu;Zhi-Ming Zhang;Inna Khazhieva;Morzherin Y. Yurievich;Nataliya P. Belskaya;Vasiliy A. Bakulev |
19 | 一类含4-甲基-1,2,3-噻二唑的α-(取代)羟基酰胺衍生物及其制备方法和用途 | 专利 | 范志金;李岳东;陈旭艳;李娟娟;房震;姬晓恬;华学文;毛武涛;宗广宁;李凤云 |
20 | Discovery and structure-activity relationship of novel diphenylthiazole derivatives as BTK inhibitor with potent activity against B cell lymphoma cell lines. | 期刊论文 | Guo Xiaofeng;Yang Dongyan;Fan Zhijin;Zhang Nailou;Zhao Bin;Huang Chun;Wang Fangjie;Ma Rongji;Meng Meng;Deng Youcai |
21 | Design, Synthesis and Biological Evaluation of Isothiazole Based 1,2,4-Trizaole Derivatives | 期刊论文 | Chen Lai;Wu Qifan;Fan Zhijin;Li Hongpeng;Li Jiwei;Hu Wenhao;Liu Xiumei;Belskaya Nataliya P;Glukhareva Tatiana;Zhao Bin |
22 | Efficient construction of bioactive trans-5(A)5(B)6(C) spirolactones via bicyclo[4.3.0] alpha-hydroxy ketones | 期刊论文 | Y. J. Zhu;J. Q. Huo;Z. J. Fan;Q. F. Wu;X. Li;S. Zhou;L. X. Xiong;T. Kalinina;T. Glukhareva |
23 | 一类含4,5-二氢噻唑醇酸酯的5-甲基-1,2,3-噻二唑衍生物及其制备方法和用途 | 专利 | 范志金;毛武涛;李娟娟;姬晓恬;华学文;宗广宁;李凤云;刘超伦;周漓轲;程胜名;房震;李岳东 |
24 | A kind of isothiazole oxime ether containing strobilurin derivatives and its preparation methods and application | 专利 | Fan Zhijin;Chen Lai;Guo Xiaofeng;Zhu Yujie;Qian Xiaolin;Ma Liuyong;Zhang Nailou;Wang Haixia;Zhang Zhiming;Xu Jinghua;Song Yinqi |
25 | 一类异噻唑肟醚甲氧基丙烯酸酯衍生物及其制备方法和用途 | 专利 | Fan Zhijin;Chen Lai;Guo Xiaofeng;Zhu Yujie;Qian Xiaolin;Ma Liuyong;Zhang Nailou;Wang Haixia;Zhang Zhiming;Xu Jinghua;Song Yinqi |
26 | Synthesis, bioactivity and mode of action of 5(A)5(B)6(C) tricyclic spirolactones as novel antiviral lead compounds | 期刊论文 | Zhu Yu Jie;Wu Qi Fan;Fan Zhi Jin;Huo Jing Qian;Zhang Jin Lin;Zhao Bin;Lai Chen;Qian Xiao Lin;Ma De Jun;Wang Da Wei |
27 | 基于氧化固醇结合蛋白的哌啶基噻唑类新农药创制研究进展 | 期刊论文 | 吴启凡;郝泽生;范志金 |
28 | 一类2位苯基取代噻唑衍生物及其制备方法和用途 | 专利 | 范志金;郭晓凤;赵斌;张乃楼;杨冬燕;吴启凡;于斌;周爽;秦忠翔 |
29 | 96%甲噻诱胺原药登记证 | 奖励 | 范志金;范谦;邱丰;殷勇;员工们 |
30 | 一类含4-甲基-1,2,3-噻二唑的甲脒衍生物及其制备方法和用途 | 专利 | 范志金;房震;陈旭艳;李娟娟;李岳东;姬晓恬;华学文;毛武涛;宗广宁;李凤云;刘超伦;周漓轲;程胜名 |
31 | A Synthetic Disaccharide Derivative of Diphyllin, TAARD, Activates Human Natural Killer Cells to Secrete Interferon-Gamma via Toll-Like Receptor-Mediated NF-kappa B and STAT3 Signaling Pathways | 期刊论文 | Yi Long;Chen Luxi;Guo Xiaofeng;Lu Ting;Wang Haixia;Ji Xiaotian;Zhang Jianying;Ren Yulin;Pan Pan;Kinghorn A Douglas;Huang Xiaohua;Wang Li Shu;Fan Zhijin;Caligiuri Michael A;Yu Jianhua |
32 | 一类含3,4-二氯异噻唑的甲氧基丙烯酸酯衍生物及其制备方法和用途 | 专利 | 范志金;杨冬燕;李正名;王海霞;郭晓凤;张乃楼;吴启凡;于斌;周爽 |
33 | 一种α-氨基丙烯酸类杀微生物剂及其制备方法和用途 | 专利 | 范志金;钱晓琳;薛景;吴傲奔;杨怀普;马刘勇;于斌;王海霞;张乃楼;吴启凡;韩岑晖;金健宇 |
34 | 一类含4,5-二氢噻唑醇酸酯的3,4-二氯异噻唑衍生物及其制备方法和用途 | 专利 | 范志金;宗广宁;李凤云;李岳东;李娟娟;姬晓恬;陈来;朱玉洁;刘超伦;程胜名 |
35 | Synthesis and biological activity of novel succinate dehydrogenase inhibitor derivatives as potent fungicide candidates | 期刊论文 | Dongyan Yang;Bin Zhao;Zhijin Fan;Bin Yu;Nailou Zhang;Zhengming Li;Yilin Zhu;Jinghui Zhou;Tatiana A. Kalinina;Tatiana V. Glukhareva |
36 | 201610185794.2 | 专利 | 范志金;朱玉洁;徐京华;宋胤奇;张秩鸣;张乃楼;王海霞;陈来;马刘勇;钱晓琳;郭晓凤 |
37 | 一类噻二唑肟醚甲氧基丙烯酸酯衍生物及其制备方法和用途 | 专利 | Fan Zhijin;Chen Lai;Zhang Zhiming;Zhang Nailou;Guo Xiaofeng;Zhu Yujie;Qian Xiaolin;Ma Liuyong;Wang Haixia;Xu Jinghua;Song Yinqi;Liang Fuqi;Tian Haifeng;Yu Maoxiang |
38 | 一类溴代六氢茚酮类化合物及其制备方法和用途 | 专利 | Fan Zhijin;Zhu Yujie;Xu Jinghua;Song Yinqi;Zhang Zhiming;Zhang Nailou;Wang Haixia;Chen Lai;Ma Liuyong;Qian Xiaolin;Guo Xiaofeng |
39 | 一类噻二唑和异噻唑酰胺类衍生物及其制备方法和用途 | 专利 | 范志金;杨冬燕;李正名;朱奕霖;周静会;郭晓凤;张乃楼;吴启凡;于斌;周爽 |
40 | 一类含氮杂环的噻唑衍生物及其制备方法和用途 | 专利 | 范志金;朱玉洁;李凤云;宗广宁;陈来;杨俊超;石凯;马刘勇;王海霞;钱晓琳;郭晓凤 |
41 | Discovery of novel piperidinyl-thiazole derivatives as broad-spectrum fungicidal candidate | 期刊论文 | Wu Qifan;Zhao Bin;Fan Zhijin;Guo Xiaofeng;Yang Dongyan;Zhang Nailou;Yu Bin;Zhou Shuang;Zhao Jiabao;Chen Fan |
42 | 一类5A5B6C三环螺环内酯衍生物及其制备方法和用途 | 专利 | 范志金;朱玉洁;陈来;周爽;郭晓凤;王海霞;于斌;张乃楼;吴启凡;杨冬燕;赵斌 |
43 | 24%甲噻·吗啉胍悬浮剂登记证 | 奖励 | 范志金;范谦;邱丰;殷勇;员工们 |
44 | 一类3,4-二氯异噻唑衍生物及其制备方法和用途 | 专利 | 陈晓燕;刘细平;范志金;梁小文;李岳东;毛武涛;李娟娟;王盾;王曙华;周立峰;姬晓恬;华学文;黄亮文 |
45 | 一类噻二唑肟醚甲氧基丙烯酸酯衍生物及其制备方法和用途 | 专利 | 范志金;陈来;张秩鸣;张乃楼;郭晓凤;朱玉洁;钱晓琳;马刘勇;王海霞;徐京华;宋胤奇;梁福起;田海丰;于茂祥 |
46 | 一类木脂素类衍生物及其制备方法和用途 | 专利 | 范志金;姬晓恬;余建华;李娟娟;华学文;宗广宁;李凤云;刘超伦;朱玉洁;陈来 |
47 | Mode of action for a new potential fungicide candidate, 3-(4-Methyl-1,2,3-thiadiazolyl)-6-trichloromethyl-[1,2,4]-triazolo-[3,4- b][1,3,4]-thiadiazole by iTRAQ | 期刊论文 | Zhao Bin;Wang Haixia;Fan Zhijin;Wu Qifan;Guo Xiaofeng;Zhang Nailou;Yang Dongyan;Yu Bin;Zhou Shuang |
48 | 一类异噻唑联噻唑衍生物及其制备方法和用途 | 专利 | 范志金;吴启凡;陈来;刘秀梅;郭晓凤;杨冬燕;张乃楼;于斌;赵斌;朱玉洁 |
49 | 一类哌啶噻唑衍生物及其制备方法和用途 | 专利 | 范志金;李凤云;张雨晴;石凯;马刘勇;郭晓凤;钱晓琳;宗广宁;朱玉洁;陈来 |
50 | 一类3,4-二氯异噻唑双酰肼类化合物及其制备方法和用途 | 专利 | 范志金;宗广宁;李岳东;李娟娟;李凤云;姬晓恬;朱玉洁;陈来;刘超伦;程胜名 |
51 | Design, synthesis and fungicidal activity of isothiazole-thiazole derivatives | 期刊论文 | Qi-Fan Wu;Bin Zhao;Zhi-Jin Fan;Jia-Bao Zhao;Xiao-Feng Guo;Dong-Yan Yang;Nai-Lou Zhang;Bin Yu;Tatiana Kalinina;Tatiana Glukhareva |
52 | 一类含氮含硫磺酰亚胺衍生物及其制备方法和用途 | 专利 | 范志金;朱玉洁;郭晓凤;陈来;钱晓琳;马刘勇;张乃楼;王海霞;裴钰;徐京华 |
53 | 一类噻唑醛肟醚类化合物及其制备方法和用途 | 专利 | 范志金;朱玉洁;郭晓凤;王海霞;李凤云;宋胤奇;徐京华;王家然;钱晓琳;马刘勇;陈来;宗广宁 |
54 | 一类杂环吗啉类衍生物及其制备方法和用途 | 专利 | 范志金;陈来;李鸿鹏;刘秀梅;赵斌;吴启凡;朱玉洁;张乃楼;于斌;杨冬燕;王海霞;郭晓凤 |
55 | 一种α-氨基丙烯酸类杀微生物剂及其制备方法和用途 | 专利 | Fan Zhijin;Qian Xiaolin;Xue Jing;Wu Aoben;Yang Huaipu;Yang Huaipu;Yu Bin;Wang Haixia;Zhang Nailou;Wu Qifan;Han Cenhui;Jin Jianyu |
56 | 一类氯代异噻唑新烟碱类化合物及其制备方法和用途 | 专利 | 范志金;宗广宁;马刘勇;张乃楼;郭晓凤;朱玉洁;陈来;钱晓琳;王海霞;张秩鸣;梁福起;田海丰 |
57 | 一类手性四氢吡啶衍生物及其制备方法和用途 | 专利 | 范志金;朱玉洁;陈来;郭晓凤;马刘勇;钱晓琳;张乃楼;王海霞;王盼盼;宋胤奇 |
58 | Synthesis, crystal structure and biological activity of 2-(1-(3-bromo-1-(3-chloropyridin-2-yl)-1H- pyrazole-5-carbonyl) piperidin-4-yl)-N-isopropyl-1,3-thiazole-4-carboxamide | 奖励 | Li Feng-Yun;Zhu Yu-Jie;Fan Zhi-Jin;Xu Jing-Hua;Guo Xiao-Feng;Zong Guang-Ning;Song Hai-Bin;Chen Lai;Song Yin-Qi;Qian Xiao-Lin;Ma Liu-Yong;Wang Jia-Ran |
59 | 一类含噻二唑杂环的新烟碱类化合物及其制备方法和用途 | 专利 | 范志金;马刘勇;宗广宁;郭晓凤;钱晓琳;朱玉洁;陈来;李凤云;李娟娟;徐京华;梁福起;田海丰;于茂祥 |
60 | 一类含二氟乙基的杂环化合物及其制备方法和用途 | 专利 | 范志金;宗广宁;马刘勇;陈来;郭晓凤;钱晓琳;裴钰;梁福起;田海丰;李吉宏;张毅超;于茂祥 |
61 | Discovery of Novel Thiazole Carboxamides as Antifungal Succinate Dehydrogenase Inhibitors | 期刊论文 | Guo Xiaofeng;Zhao Bin;Fan Zhijin;Yan Dongyan;Zhang Nailou;Wu Qifan;Yu Bin;Zhou Shuang;Kalinina Tatiana A;Belskaya Nataliya P |