新型自旋标记喹啉类拓扑异构酶I抑制剂的设计合成及其生物活性研究
序号 | 标题 | 类型 | 作者 |
---|---|---|---|
1 | Design and synthesis of novel 7-[(N-substitutedthioureidopiperazinyl)- methyl]-camptothecin derivatives as potential cytotoxic agents | 期刊论文 | Zi-Long Song;Guan-Zhou Yang;Jun-Cai Li;Ying-Qian Liu;Chen-Jie Yang;Masuo Goto;Zhi-Jun Zhang;Susan L. Morris-Natschke;Hua Liu;Kuo- Hsiung Lee |
2 | 一种7-乙基-10-氟-喜树碱-20-肉桂酯类化合物、制备方法和用途 | 专利 | 刘映前;杨程杰;Raymond Kobla Lawoe;李俊采;张晓帅;徐小山;杨冠洲;陈诚;张君香 |
3 | 一种6H-苯并吡喃并[3,4-b]喹啉类化合物及其制备方法和用途 | 专利 | 刘映前;徐传瑞;高建梅;杨程杰;白银鹏;张智军;李海欣;赵文斌 |
4 | 一种喜树碱20-位修饰的磺酰胺类化合物及其制备方法和用途 | 专利 | 刘映前;雷蒙·科布拉·劳威;杨程杰;宋子龙;李虎;高建梅 |
5 | 一种氟化苯并萘啶酮类衍生物、制备方法及用途 | 专利 | 刘映前;徐小山;李俊采;陈诚;张君香;张晓帅;杨冠洲;杨程杰 |
6 | Biologically active indolizidine alkaloids | 期刊论文 | Junmin Zhang;Susan L. Morris‐Natschke;Di Ma;Xiao‐Fei Shang;Chen‐Jie Yang;Ying‐Qian Liu;Kuo‐Hsiung Lee |
7 | Biologically active quinoline and quinazoline alkaloids part II | 期刊论文 | Shang Xiao Fei;Morris Natschke Susan L;Yang Guan Zhou;Liu Ying Qian;Guo Xiao;Xu Xiao Shan;Goto Masuo;Li Jun Cai;Zhang Ji Yu;Lee Kuo Hsiung |
8 | 一种稳定氮 氧自由基标记的茚并异喹啉衍生物、制备方法及用途 | 专利 | 刘映前;徐小山; 张晓帅;杨冠洲;刘华;高建梅;陈诚;张君香 |
9 | 以天然源喜树碱为先导的抗肿瘤药物的设计合成与新药创制研究 | 奖励 | 刘映前;田瑄;杨柳;王美娟;赵永龙;赵晓博 |
10 | Design, synthesis and potent cytotoxic activity of novel 7-(N-[(substituted-sulfonyl)piperazinyl]-methyl)-camptothecin derivatives | 期刊论文 | Zhu Gao-Xiang;Cheng Pi-Le;Goto Masuo;Zhang Na;Morris-Natschke Susan L.;Hsieh Kan-Yen;Yang Guan-Zhou;Yang Qian-Ru;Liu Ying-Qian;Chen Hai-Le;Zhang Xiao-Shuai;Lee Kuo-Hsiung |
11 | Design, semisynthesis and potent cytotoxic activity of novel 10-fluorocamptothecin derivatives | 期刊论文 | Yang Cheng Jie;Song Zi Long;Goto Masuo;Hsu Pei Ling;Zhang Xiao Shuai;Yang Qian Ru;Liu Ying Qian;Wang Mei Juan;Morris Natschke Susan L;Shang Xiao Fei;Lee Kuo Hsiung |
12 | 一种喜树碱20-位修饰的磺酰脲类化合物及其制备方法和用途 | 专利 | 刘映前;高建梅;杨程杰;李虎;宋子龙;雷蒙·科布拉·劳威 |
13 | Design, synthesis, and cytotoxic activity of novel 7-substituted camptothecin derivatives incorporating piperazinyl-sulfonylamidine moieties | 期刊论文 | Yang Cheng Jie;Song Zi Long;Goto Masuo;Liu Ying Qian;Hsieh Kan Yen;Morris Natschke Susan L;Zhao Yong Long;Zhang Jun Xiang;Lee Kuo Hsiung |
14 | Biologically active isoquinoline alkaloids covering 2014–2018 | 期刊论文 | Xiao‐Fei Shang;Cheng‐Jie Yang;Susan L. Morris‐Natschke;Jun‐Cai Li;Xiao‐Dan Yin1;Ying‐Qian Liu;Xiao Guo;Jing‐Wen Peng;Masuo Goto;Ji‐Yu Zhang;Kuo‐Hsiung Lee |
15 | Nanocrystals of a new camptothecin derivative WCN-21 enhance its solubility and efficacy | 期刊论文 | You Jia;Chen Yuyuan;Alsayeh Zubaeda M. Mohamed;Shen Xingyu;Li Chun;Zhao Pengxuan;Chen Fei;Liu Yingqian;Xu Chuanrui |
16 | Design, synthesis and antineoplastic activity of novel 20(S)- acylthiourea derivatives of camptothecin | 期刊论文 | Cheng-Jie Yang;Bin Li;Zhi-Jun Zhang;Jian-Mei Gao;Mei-Juan Wang;Xiao-Bo Zhao;Zi-Long Song;Ying-Qian Liu;Hu Li;Yuyuan Chen;Kuo-Hsiung Lee;Susan L. Morris-Natschke;Chuanrui Xu |
17 | 一种9-位哌嗪磺酰胺-10-羟基喜树碱类化合物及其制备方法和在抗肿瘤中的用途 | 专利 | 刘映前;陈海乐;杨程杰;雷蒙·科布拉·劳威;李虎;高建梅 |
18 | Biologically active quinoline and quinazoline alkaloids part I | 期刊论文 | Shang Xiao-Fei;Morris-Natschke Susan L.;Liu Ying-Qian;Guo Xiao;Xu Xiao-Shan;Goto Masuo;Li Jun-Cai;Yang Guan-Zhou;Lee Kuo-Hsiung |